What is Superdrol?

There is a huge possibility that Superdrol is on the list of prohormones that you have considered to help you with serious size, strength and mass gains.

But if you’re still a bit unsure about choosing this one, make sure you follow along to find out more about this successful prohormone that took the bodybuilding world by storm in the last decade.

Let’s start off by clarifying one popular misconception about this prohormone. Superdrol isn’t an ingredient that makes this prohormone but is actually the name of the brand that marketed it when it was released in 2015 by Designer Supplements LLC.  The name Superdrol is basically a combination of “Super” and “Anadrol” where Anadrol is an oral steroid that was known as one the most powerful mass builder in history.

The active compound in this prohormone is methasterone also known as methasteron and methyldrostanolone. Its systematic IUPAC name is 17β-Hydroxy-2α,17α-dimethyl-5α-androstane-3-one. The half-life of this prohormone is 6-8 hours.  Superdrol became a legend in the bodybuilding world due to its speedy results in terms of significant hard and dry gains within a few weeks of usage. Superdrol gained huge success in a very short period of time.  Many of its users were happy with the results and reported to gain 20-30 pounds of muscle mass within 4 weeks of usage.

Besides providing a considerable boost in size and mass, this dihydrotestosterone or DHT-derived prohormone also has the ability to take strength levels up a notch. The users of this compound claim that they were able to increase their overall lifts by as much as 20 to 25 percent in just the second week of their cycle with this compound.

Superdrol’s power and intensity come from the fact that it is quite similar to Masteron, a different type of anabolic steroid, but without the ester chain that the latter flaunts in its chemical structure. It works by optimizing the body’s ability to retain nitrogen and its synthesis of protein, which results not just in gains in size, mass, strength, and endurance, but also the speed muscles recover after going through a grueling workout.

Plus its androgenic activity in the body is much lower compared to its prohormone counterparts. This means that Superdrol doesn’t put you at risk of experiencing increased hair loss or hair growth as well as bouts of acne when you use it compared to other anabolic steroids. Also, it isn’t necessary to use an anti-estrogen when cycling with this compound.

During the time when Superdrol was freely available on the shelves, this orally ingested prohormone was considered as a crucial bulking, cutting and recovery agent that yielded quick results without having to do anything with needles. This was the biggest reason why it earned a lot of loyal followers worldwide.

Superdrol is basically a type of C17-aa anabolic steroid and can be toxic to the liver, especially when used without the proper on-cycle support and post cycle therapy. Clinical researchers emphasize that cycling with this prohormone can trigger the values of liver enzymes to surge, which causes stress and can lead to health issues if not given the right attention it deserves.

Now while Superdrol was taking the bodybuilding world by storm, it was banned by the U.S. Food and Drug Administration (FDA) in 2006, which forced its manufacture and distribution to halt. However, the ban did not stop the production and sale of the methasterone compound in both legal consumer over-the-counter market and underground channels.

The FDA cracked down on this further by classifying the prohormone as a Schedule III controlled substance, along with other anabolic steroids, in August 29, 2012. There are still Superdrol “clones” that you can get your hands on these days.

After this prohormone’s ban took effect in 2012, many of its users picked Dymethazine as an alternative. Dymethazine is made up of two Superdrol molecules that are kept together by a single nitrogen atom. It was spared from the ban because it had an entirely different hormonal structure.

Although Superdrol was launched in the market as a “designer steroid” in 2005, its active compound ‘methasterone’ had been formulated long ago in 1956 by the Syntex Corporation while developing a compound that staves off tumors.

In addition to its anti-tumor properties, the compound was also recognized for its oral bioavailability and high anabolic vs. androgenic ratio of 20.  A scientific article written in 1959 describes methasterone as an orally active potent anabolic agent with weak androgenic effect.

However, methasterone did not fully become a prescription drug even with its proven attributes. The Syntex Corporation instead focused on developing a non-17α-alkylated counterpart of this compound called drostanolone and eventually released it in the market as Masteron. It wasn’t until 2005 that methasterone – in the form of Superdrol – hit the shelves as a dietary supplement, which didn’t take long for it to become a huge success.


If you’re planning to integrate Superdrol in your bodybuilding checklist, here are the benefits that you will be in for:

  • It helps boost size and mass gains
  • It increases overall strength levels
  • It boosts nitrogen retention and protein synthesis
  • It can be used without an anti-estrogen.
  • No serious estrogenic effects like increased facial hair in women, enlarged breasts in men, and depression etc. This is one of the safest options available in the market when it comes to body-building steroids. Since the prohormone is not converted to estrogen, this supplement comes without the negative side effects associated with estrogen.
  • It doesn’t have as much androgenic activity compared to its counterparts
  • It can yield up to 30 pounds of lean muscle in 4 weeks
  • It acts really fast. It considerably improves your body’s protein synthesis leading to increased muscle growth.   In this way, it helps you gain muscle mass quickly.


It is very important to take note that small doses of Superdrol should be taken during the start of a cycle. Experienced users highly recommend that you begin with a daily dose of 10mg for the first week and increase your dosage to 20mg in the second and third week. It’s necessary to take Superdrol daily with food. If you are very tolerant of this compound, you can bump up to 40mg in the fourth week.

Moreover, experienced Superdrol users suggest that this compound stacks quite well with most anabolic steroids. Stacking some form of testosterone with this prohormone considerably helps you in achieving your cutting and bulking goals. Trenbolone is highly recommended with Superdrol when cutting, while Nandrolone is a nice choice to stack with this compound during a bulking phase.

The user should undergo proper post cycle therapy in the succeeding fifth to the eighth week. PCT helps in restoring your organs’ health and brings your hormone levels back to normal.

It helps you maintain your gains and restores your overall health. As you know, when we run a prohormone, our body stops producing its natural hormones. What a post cycle therapy does is that it restores your body to its natural state thereby leading it to produce hormones at natural levels again. In this way, it brings your hormones to natural levels and saves you from the unpleasant side effects that could otherwise turn up.

Going into more detail about “how” a PCT normalizes your hormone levels, what it basically does is that it controls the production of estrogen (the hormone responsible for almost all the trouble) and boosts the production of testosterone (the hormone that eliminates excess body fat, helps you gain and maintain muscle mass in your body, strengthens your heart and provides many other benefits).

We would recommend cycling on Selective estrogen receptor modulator (SERM) a day after completion of Superdrol cycle. Clomid, Toremifene, and Nolva are commonly chosen by people. After reviewing all three, we would personally go with Clomid.  It is the fastest way of restoring the production of testosterone. Remember that testosterone production is vital for retaining gains in post-cycle therapy. However, Nolva is a better choice if your first priority is estrogen control.

Side Effects

Although Superdrol has lower androgenic levels compared to other prohormones in the market, you can still be vulnerable to the following side effects when you cycle with it:

  • It can cause a spike in blood pressure and bad cholesterol levels
  • It can place the body in a low testosterone state
  • It can be toxic to the liver in absence of proper support and precautions

A Quick Rundown on a Superdrol Cycle

Perhaps the most important guideline that you should keep in mind to make your cycle with Superdrol as successful as possible is having an idea about the right dosage to get you on track to achieve your goals. Here is a quick guide that you can use to kick off your cycle with this prohormone.

Superdrol Reviews

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Final Verdict

Considering all the pros and cons of Superdrol, we can certainly say that it is one of the best prohormones available these days. It provides its users with a long range of benefits s without the negative side effects that usually come with other steroids. This anabolic prohormone is an all-rounder as it increases muscle mass and strength levels along with speeding up protein synthesis and recovery process.

This anabolic prohormone definitely deserves to be in your bodybuilding arsenal!

However, make sure that you’re taking your doses in the right amount at the right time. Also, it is highly recommended to go for an on-cycle support and a post-cycle therapy to be on the safe side. You surely don’t want to compromise on your health, do you? An on-cycle support will curtail the potential side effects of this prohormone whereas PCT will restore your body’s overall health and help you maintain your gains.


You will most probably test positive while using 1-Andro during anabolic steroid testing due to the excretion of metabolites from 1-Testosterone. Make sure to speak with the drug administer if you have any worries before taking 1-Androsterone.

Yes, you need to have cycle support and PCT when running 1-Andro to make sure optimal health and avoid unwanted side effects. Supplements to combat hair loss added to your cycle will also help, such as Infinity Hair.

Post cycle therapy is necessary as this assists in repairing natural testosterone production at the end of your cycle. Watch the video below to help you ace your PCT to avoid losing those hard-earned gains.

Yes, it is possible to retain your gains after completing the cycle.  In order to do that, you should take Nolvadex. This will help you lose bloat that has resulted from water retention. Taking nitrous based compounds and creatine is also a good choice to retain your gains.

We have come across many people who want to start another cycle right after completing their PCT. Superdrol surely gives amazing results, but it is important to understand that you have a life apart from bodybuilding and you don’t want to lose that, right?  So we would recommend you to please take a two months break before starting another cycle, otherwise, your liver will be severely damaged.

Superdrol has a half-life of 6-8 hours, therefore, it is recommended to take it every 6 to 8 hours. Different people have varying answers to this question. However, the majority says that the first dose should be taken in the morning with plenty of water with an empty stomach. This means that you should not eat anything before taking this dose.  The best time for next dose is with your pre-workout meal with a good amount of healthy fats like peanut butter or fish oils.

Superdrol has a heavy influence on your lipid profile. Eating a fat or carb-rich meal can help you out here to some extent.  People have mixed opinions on this. Taking a Superdrol dose before a workout increases your strength during workout sessions.

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